| Delineating the role of cooperativity in the design of potent PROTACs for BTK A Zorba, C Nguyen, Y Xu, J Starr, K Borzilleri, J Smith, H Zhu, KA Farley, ... Proceedings of the National Academy of Sciences 115 (31), E7285-E7292, 2018 | 319 | 2018 |
| A New Resistance Gene, linB, Conferring Resistance to Lincosamides by Nucleotidylation in Enterococcus faecium HM1025 B Bozdogan, L Berrezouga, MS Kuo, DA Yurek, KA Farley, BJ Stockman, ... Antimicrobial agents and chemotherapy 43 (4), 925-929, 1999 | 239 | 1999 |
| Discovery of cytotoxic dolastatin 10 analogues with N-terminal modifications A Maderna, M Doroski, C Subramanyam, A Porte, CA Leverett, ... Journal of medicinal chemistry 57 (24), 10527-10543, 2014 | 140 | 2014 |
| Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance AC Rand, SSF Leung, H Eng, CJ Rotter, R Sharma, AS Kalgutkar, ... MedChemComm 3 (10), 1282-1289, 2012 | 136 | 2012 |
| Integrating intramolecular hydrogen bonding (IMHB) considerations in drug discovery using ΔlogP as a tool M Shalaeva, G Caron, YA Abramov, TN O’Connell, MS Plummer, ... Journal of medicinal chemistry 56 (12), 4870-4879, 2013 | 95 | 2013 |
| Non-uniform sampling for all: more NMR spectral quality, less measurement time F Delaglio, GS Walker, KA Farley, R Sharma, JC Hoch, LW Arbogast, ... American pharmaceutical review 20 (4), 2017 | 68 | 2017 |
| Methods for creating a compound library and identifying lead chemical templates and ligands for target molecules BJ Stockman, KA Farley, C Dalvit US Patent 6,677,160, 2004 | 61 | 2004 |
| Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections TV Magee, SL Ripp, B Li, RA Buzon, L Chupak, TJ Dougherty, ... Journal of medicinal chemistry 52 (23), 7446-7457, 2009 | 58 | 2009 |
| A new and useful method for the macrocyclization of linear peptides AT Londregan, KA Farley, C Limberakis, PB Mullins, DW Piotrowski Organic letters 14 (11), 2890-2893, 2012 | 54 | 2012 |
| Screening of compound libraries for protein binding using flow-injection nuclear magnetic resonance spectroscopy BJ Stockman, KA Farley, DT Angwin Methods in enzymology 338, 230-246, 2002 | 41 | 2002 |
| Increased HMBC sensitivity for correlating poorly resolved proton multiplets to carbon-13 using selective or semi-selective pulses A Bax, KA Farley, GS Walker Journal of Magnetic Resonance, Series A 119 (1), 134-138, 1996 | 41 | 1996 |
| Design and evaluation of a 2-(2, 3, 6-trifluorophenyl) acetamide derivative as an agonist of the GPR119 receptor V Mascitti, BD Stevens, C Choi, KF McClure, CRW Guimarães, KA Farley, ... Bioorganic & medicinal chemistry letters 21 (5), 1306-1309, 2011 | 33 | 2011 |
| Complete spectroscopic structural characterization of novobiocin, isonovobiocin, decarbamylnovobiocin, 2″‐(o‐Carbamyl)novobiocin, and novobiocin‐2″,3 … FW Crow, WK Duholke, CE Hadden, RF Smith, TJ Thamann, BD Kaluzny, ... Journal of heterocyclic chemistry 36 (2), 365-370, 1999 | 33 | 1999 |
| Macrocyclizations for medicinal chemistry: Synthesis of druglike macrocycles by high-concentration Ullmann coupling JC Collins, KA Farley, C Limberakis, S Liras, D Price, K James The Journal of Organic Chemistry 77 (24), 11079-11090, 2012 | 31 | 2012 |
| Hierarchical mesoporous bio-polymer/silica composites co-templated by trimethyl chitosan and a surfactant for controlled drug delivery VK Rana, SS Park, S Parambadath, MJ Kim, SH Kim, S Mishra, RP Singh, ... MedChemComm 2 (12), 1162-1166, 2011 | 31 | 2011 |
| Long‐range two‐dimensional 1H–15N heteronuclear shift correlation at natural abundance using GHNMQC. A study of the reverse transcriptase inhibitor delavirdine KA Farley, GS Walker, GE Martin Magnetic resonance in chemistry 35 (10), 671-679, 1997 | 27 | 1997 |
| Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis KA Farley, Y Che, A Navarro-Vázquez, C Limberakis, D Anderson, J Yan, ... The Journal of Organic Chemistry 84 (8), 4803-4813, 2019 | 26 | 2019 |
| Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue DA Price, H Eng, KA Farley, GH Goetz, Y Huang, Z Jiao, AS Kalgutkar, ... Organic & Biomolecular Chemistry 15 (12), 2501-2506, 2017 | 23 | 2017 |
| The synthesis of C-13 functionalized pleuromutilins via C–H amidation and subsequent novel rearrangement product DP Uccello, SM Miller, NA Dieterich, AF Stepan, SW Chung, KA Farley, ... Tetrahedron letters 52 (33), 4247-4251, 2011 | 23 | 2011 |
| Utilizing on‐and off‐line monitoring tools to follow a kinetic resolution step during flow synthesis KA Farley, U Reilly, DP Anderson, BP Boscoe, MW Bundesmann, ... Magnetic Resonance in Chemistry 55 (4), 348-354, 2017 | 21 | 2017 |
Brian StockmanAdelphi UniversityDirección de correo verificada de adelphi.edu
