Timothy A Hill
Timothy A Hill
Senior Reserch Officer, University of Queensland
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Constraining cyclic peptides to mimic protein structure motifs
TA Hill, NE Shepherd, F Diness, DP Fairlie
Angewandte Chemie International Edition 53 (48), 13020-13041, 2014
A novel class of anticancer compounds targets the actin cytoskeleton in tumor cells
JR Stehn, NK Haass, T Bonello, M Desouza, G Kottyan, H Treutlein, ...
Cancer research 73 (16), 5169-5182, 2013
Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency
RS Harrison, NE Shepherd, HN Hoang, G Ruiz-Gómez, TA Hill, ...
Proceedings of the National Academy of Sciences 107 (26), 11686-11691, 2010
Comparative α‐Helicity of cyclic pentapeptides in water
AD De Araujo, HN Hoang, WM Kok, F Diness, P Gupta, TA Hill, RW Driver, ...
Angewandte Chemie International Edition 53 (27), 6965-6969, 2014
Inhibition of Dynamin Mediated Endocytosis by the DynolesSynthesis and Functional Activity of a Family of Indoles
TA Hill, CP Gordon, AB McGeachie, B Venn-Brown, LR Odell, N Chau, ...
Journal of medicinal chemistry 52 (12), 3762-3773, 2009
Systemic delivery of peptides by the oral route: Formulation and medicinal chemistry approaches
DJ Brayden, TA Hill, DP Fairlie, S Maher, RJ Mrsny
Advanced drug delivery reviews 157, 2-36, 2020
Improving on nature: making a cyclic heptapeptide orally bioavailable
DS Nielsen, HN Hoang, RJ Lohman, TA Hill, AJ Lucke, DJ Craik, ...
Angewandte Chemie International Edition 53 (45), 12059-12063, 2014
Norcantharimides, synthesis and anticancer activity: Synthesis of new norcantharidin analogues and their anticancer evaluation
TA Hill, SG Stewart, SP Ackland, J Gilbert, B Sauer, JA Sakoff, ...
Bioorganic & medicinal chemistry 15 (18), 6126-6134, 2007
Heterocyclic substituted cantharidin and norcantharidin analogues—synthesis, protein phosphatase (1 and 2A) inhibition, and anti-cancer activity
TA Hill, SG Stewart, B Sauer, J Gilbert, SP Ackland, JA Sakoff, ...
Bioorganic & medicinal chemistry letters 17 (12), 3392-3397, 2007
Green chemistry approaches to the Knoevenagel condensation: comparison of ethanol, water and solvent free (dry grind) approaches
A McCluskey, PJ Robinson, T Hill, JL Scott, JK Edwards
Tetrahedron letters 43 (17), 3117-3120, 2002
Update 1 of: Beta-Strand Mimetics
Wendy A. Loughlin, Joel D. A. Tyndall, Matthew P. Glenn,Timothy A. Hill ...
Chemical Reviews 110 (6), PR32-PR69, 2010
Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins
T Hill, LR Odell, JK Edwards, ME Graham, AB McGeachie, J Rusak, ...
Journal of medicinal chemistry 48 (24), 7781-7788, 2005
Norcantharidin analogues: synthesis, anticancer activity and protein phosphatase 1 and 2A inhibition
TA Hill, SG Stewart, CP Gordon, SP Ackland, J Gilbert, B Sauer, JA Sakoff, ...
ChemMedChem: Chemistry Enabling Drug Discovery 3 (12), 1878-1892, 2008
Flexibility versus rigidity for orally bioavailable cyclic hexapeptides
DS Nielsen, RJ Lohman, HN Hoang, TA Hill, A Jones, AJ Lucke, ...
ChemBioChem 16 (16), 2289-2293, 2015
Crystal structures of protein-bound cyclic peptides
AK Malde, TA Hill, A Iyer, DP Fairlie
Chemical Reviews 119 (17), 9861-9914, 2019
Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity
TA Hill, LR Odell, A Quan, R Abagyan, G Ferguson, PJ Robinson, ...
Bioorganic & Medicinal Chemistry Letters 14 (12), 3275-3278, 2004
Cyclic Penta- and Hexaleucine Peptides without N-Methylation Are Orally Absorbed
TA Hill, RJ Lohman, HN Hoang, DS Nielsen, CCG Scully, WM Kok, L Liu, ...
ACS medicinal chemistry letters 5 (10), 1148-1151, 2014
Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis
TA Hill, A Mariana, CP Gordon, LR Odell, MJ Robertson, AB McGeachie, ...
Journal of medicinal chemistry 53 (10), 4094-4102, 2010
Fixierung cyclischer Peptide: Mimetika von Proteinstrukturmotiven
TA Hill, NE Shepherd, F Diness, DP Fairlie
Angewandte Chemie 126 (48), 13234-13257, 2014
Truncated and helix-constrained peptides with high affinity and specificity for the cFos coiled-coil of AP-1
T Rao, G Ruiz-Gómez, TA Hill, HN Hoang, DP Fairlie, JM Mason
PLoS One 8 (3), e59415, 2013
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